Category: steroid powder canada


When is The Right Age to Start Using Steroids


This is an important question about steroids. If you’re talking about or studying steroids, you’re definitely going to have this problem, like your age and weight. Age has a lot to do with steroids for a couple of different reasons.

Steroids for young

It’s certainly not the right age to take steroids, but it’s certainly not the right age for young people. Side effects of steroid use can be very effective in young people.

Steroid bodybuilders

In general, bodybuilders use steroids to build muscle and increase the number of free hormones in the body. All the anabolic products are derivatives of testosterone, with slight molecular changes. These steroids will do you a lot of good. Steroids play an important role in athletic recovery, and they also help bodybuilders gain more weight. But I can say that without steroids, bodybuilders can gain lean muscle mass through exercise, shake off body fat and muscle tension, and allow muscle growth to take days. This will lead to slow growth. So the only difference is, if you use steroids, you get explosive growth, you can just take a few days off.

Middle-aged steroids

Steroids are dangerous for middle-aged and young people alike. As I said before, young people are too young to use this. Middle-aged people wanted to look healthier, so they started using anabolic steroids. Steroids are used to improve their muscle growth and athletic performance, which they believe is a way to recapture their youth. Studies show that many middle-aged men are taking steroids to fight weight gain and rekindle their libido. There is no doubt that steroids promote the production of red blood cells, increase the oxygen supply to muscles, increase endurance, and help thin muscle matter to be produced, thus helping them. Steroids give them more energy and muscle, but behind these benefits is the fact that as the body grows, steroid injections speed up cognitive, physical and sexual decline.

Effects of steroids on middle-aged men

Steroid use can cause them to suffer long-term physical effects such as testicular atrophy, penis problems, painful urination, and breast development.

Now they add memory loss to the list. People who use steroids forget what they are going to do in the future and can’t recall memories of the past. The results showed that those who used steroids had significantly worse memory and mental executive function than those who did not.

Steroids give your body its highest levels of hormones. This is a side effect associated with testosterone. Using them can help you train harder and give you more energy, but if you stop using them, it can take years to recover, which can be very dangerous.

Conclusion

All I can say is that there is no right age to use steroids. If you want to look healthy, build muscle or have more energy, just get it through your diet and exercise. These things will definitely help you reach your goals and give you your greatest natural potential. Because your body needs to be healthy and strong to use these steroids. When you reach a point where no amount of diet or exercise can help you gain more muscle or lose more fat, you can start adding steroids at the prescribed dose. So you should start with low doses because when it comes to steroids, it’s not good to eat more. Anything in excess is harmful to us.

 


Steroid Use


Here is a self-report of a steroid-using bodybuilder. The article is written in first-person narratives. Here we go…

I was 19 and though I had been lifting weights diligently for at least 3 years, I wasn’t anyone that you’d look at and say “there’s a bodybuilder.” I was 6 feet tall and around 160 pounds. I figure I had put on around ten pounds of muscle that I wouldn’t have had without the three years of weightlifting.

After, I joined the Air Force and got stationed at Edwards AFB in Southern California in August 1984. I turned 19 five months before that. I didn’t wait long to go see the famous steroid doctor to the stars and professional bodybuilders, Dr. Kerr, in San Gabriel. Other than a guy known as the Steroid Guru who wrote The Underground Steroid Handbook, Dan Duchaine, this Dr. Kerr was the most famous expert on the subject.

This was back when steroids weren’t a scheduled controlled substance. You could go to a doctor and tell him you wanted to take them solely for the purpose of gaining muscle, strength or for bodybuilding and the doctor could legally prescribe them to you. That’s what I did. Dr. Kerr took some blood for blood tests and prescribed Anadrol-50 oral tablet steroids for me. One tablet per day.

It seemed amazing to me then that I could just add this tiny little pill to my breakfast and I would get big. But I had read quite a bit and firmly believed it to be true. In three months I weighed over 180. Another 3 months and I was around 200. I was bursting out of my uniform. And I was strong, really, really strong.

I stuck with Dr. Kerr’s prescription for six months He had me go 6 weeks on, 6 weeks off, repeat. And I started to get the look that other steroid users recognized as “in the club” and they opened up to me about better drugs, safer ones, how to deal with side effects, etc..

The one problem with the 6 on 6 off and the really strong oral Anadrol-50, was my weight would fluctuate like crazy. When I took the 6 weeks off, by the end I would lose 2/3 to 3/4 of the weight I had gained. It was because that drug put a lot of water in my muscles. So I wanted something that was supposed to be more permanent and would not cause water retention.

After six months with Dr. Kerr I “graduated” to taking trips to Tijuana pharmacies for the favorite steroid of Arnold, Primobolan. It was a BIG step as this would require injecting myself. Primobolan was considered one of the safest, if not the safest of all steroids and pretty weak. But to my thinking at the time, if it was Arnold’s favorite, there’s gotta be something to it.

For the next couple of years, I used Primobolan and built up to a really solid and well proportioned 225ish. It worked just like I expected. Slower but steady progress. And when I took a 6-week break I would only lose about 10 to 20 percent of what I gained. I stretched out my cycles to 12 weeks with a taper up, in the beginning, then 6 weeks at a set amount, then 6 weeks tapering off. Then a six-week break, repeat. I steadily gained a pound or two a month. I’d put on 10–15 pounds or so in 3 months and then lose less than 5 when on a break. It was a steady increase. Nice workouts, felt great, didn’t draw much attention to myself by having my weight yo-yo as it did with the AD-50.

I remember back when all the experts and doctors, or most anyway, would swear that steroids don’t work. Even Arnold said he “only took them the last month or so before a contest to not lose his muscle as he dieted down.” I read a book by Rick Wayne called Muscle Wars and he detailed how Arnold took shocking amounts of steroids starting in his teens. There were lots of people around him who knew this and told Wayne. The bottom line is they work and they work great. It’s too bad such a stigma has been attached to them. But it’s getting better. There are TRT clinics everywhere now helping men slow down the aging process. Speaking of that have you noticed how many older Hollywood actors who were never really known for their physiques suddenly have bodies that rival Sylvester Stallone’s in the Rocky movies? Check out Sean Penn in “The First,” and Josh Brolin in the Sicaro sequel. That’s TRT.

That was probably way more than you expected. Any other questions, feel free to ask away.


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Dianabol bodybuilding

Dianabol is the brand name of methandienone or methandrostenolone. It was used to treat hypogonadism as early as 1955. Bodybuilders began to use Dianabol after it was found to have high anabolic activity. They can gain a lot of lean muscle in a short time. Its power also increased rapidly.

Building physical strength and endurance are one of the ultimate goals of many men and even women. This desire can arise for a variety of reasons, from sports to personal fitness. Whatever the reason, you’ll need some help getting there faster. That’s why I’m introducing anabolic and androgen steroids, Dianabol. Also known as Dbol.

Dianabol effects

Dianabol is a very effective fertilizer during low season. After a few weeks, you’ll gain 20 pounds, which is great for bodybuilders. You can also pair it with a protein-rich diet for higher performance.

This makes it one of the most powerful fitness steroids on the market today. But not all athletes are in the business of gaining weight, so other non-weight-gaining steroids may be needed. These athletes can rely on steroids like Winstrol, which do not cause weight gain.

Dianabol is also very effective as a weight loss agent during weight lifting or training cycles. But many builders seem to prefer cutting under other steroids because Dianabol has a less protective effect on lean tissue.

How to use Dianabol

To reduce the risk of physical deterioration, you must use Dianabol moderately. Your body size may determine the daily dose. A moderate daily dose should be between 30 and 50 milligrams.

More than that means more risk to the body. The recommended dose is 15 to 25 milligrams, and even at this low dose, you can get good results. This does put less pressure on the body.

With a half-life of about 3 to 5 hours, the recommended dose can be divided into two doses and taken over a distance of about 5 hours. It is recommended for people who will need it in a longer period of competition or hard training.

Dianabol reviews

Dbol is actually called Methandienone, but no one actually calls it that. Bodybuilders began to use Dianabol after it was found to have high anabolic activity. They can gain a lot of lean muscle in a short time. Its power also increased rapidly.


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What is the use of Proviron?

Proviron is used to replace testosterone in men with hypogonadism. Hypogonadism in men means the body cannot produce enough testosterone.

Testosterone is a natural male hormone, called androgen, that controls normal sexual development in men.

Testosterone is essential for the development and maintenance of the male reproductive organs and for other male characteristics such as hair growth, a deep voice, sexual arousal, muscle mass, and body fat distribution.

Proviron is only available for male patients.

Proviron PCT

In the fitness world, the use of Proviron in post-cycle therapy has many inconsistencies. So we go back to the old school days when there was no SERM and men needed help in this area so Proviron was used. Today, Proviron is no longer needed for PCT, thanks to available supplements and complementary drugs. Although Proviron does not have the inhibitory effect of other compounds (Proviron, after all, is used in Europe as a fertility drug), it is still mildly inhibitory and can be counterproductive when used in PCT or bridging therapy. Therefore, there are now better options for PCT.

Proviron uses

The first is the result of its structure. It has a reduced 5-alpha, which prevents it from forming estrogen, but it has a much higher affinity for aromatase, the enzyme that converts testosterone to estrogen. This means that when administered with testosterone or another aromatase compound, it prevents the accumulation of estrogen because it binds tightly to the aromatase enzyme, preventing these steroids from interacting with it to form estrogen. Therefore, the use of Proviron has great benefits, can reduce the side effects of estrogen and water retention with other steroids noted, and thus still helps to provide the majority of lean benefits. It has also been suggested that it may reduce the actual estrogen receptor making it doubly effective at reducing circulating estrogen levels.

A second use is to increase the potency of testosterone. Normal physiological levels of testosterone in the body are mostly inactive. Up to 97% or 98% of testosterone binds to two proteins, sex hormone binding globulin (SHBG) and albumin. In this case, testosterone is largely inactive. However, like aromatase, DHT has a higher affinity for these proteins than testosterone. Therefore, when given at the same time, mesterolone will attach to SHBG and albumin, leaving more free testosterone to mediate anabolic activities such as protein synthesis. Another way to help increase revenue. This is another part of the equation that makes itself ineffective because binding to these proteins will make it no problem at the androgen receptor.

Third, in the pre-competition stage, the addition of steroids to increase the apparent hardness and muscle density. This may be because it reduces circulating estrogen, or it may be because of the down-regulation of estrogen receptors in muscle tissue, which reduces the overall amount of water in the body, makes users look thinner and has a visual effect of “harder” muscles with more cuts and stripes. Provence is often used as a last minute secret by many bodybuilders, actors and models alike, to keep in top shape day in and day out when needed. Like drostanolone, another methylated DHT compound, mesterolone is particularly effective at achieving this goal.

Finally, Proviron is used in the cycle of certain hormones, such as nandrolone, that are noticeably lacking in androgenic properties, or possibly a 5– the reduced hormone that does not have the same affinity as DHT. This compound, especially trenbolone, nandrolone, and others, has been found to reduce libido. Restricting athletes’ sexual performance is the logical outcome. DHT plays a key role in this process, so its use with these steroids can alleviate or alleviate the annoying side effects. Proviron is usually prescribed to people with low testosterone levels or chronic impotence. It is not considered a powerful anabolic hormone, but it works just as well, if not better than other anabolic steroids, making it a popular medical practice because of its lower chance of abuse.

Proviron reviews

Mesterolone is popular because it has few side effects on men. At high doses, it can cause some masculine symptoms in women. However, due to the high inactivation and predestination (albumin, SHBG, 3bHSD, aromatase) in the system, if not all cannot reach the androgen receptor, it will lead to anabolic effects, but also have side effects. So it’s relatively safe. Use 25 to 250 milligrams daily with no side effects. For the four conditions mentioned above, 50 milligrams per day is usually enough to be effective, so there is no need to drink more. Not as some suggest or believe,


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What is Testosterone Propionate?

It is a very important compound of testosterone. Testosterone propionate is an oil-based steroid containing propionate. Testosterone propionate is released the fastest, but it must be injected daily for good results. Another advantage of this compound is that it can be easily controlled to prevent any side effects. It’s different with testosterone enanthate, enanthate role is much slower than propionate, propionate needs more frequent injections in order to ensure stable blood concentration.

How to order Testosterone Propionate online?

Once you’ve selected the testosterone propionate product, you just add it to your shopping list. Anyone can order testosterone propionate through this website at sale@getraws.com: this means we are happy to send your order to any address in the United States, United Kingdom, Canada, Australia, Europe or Africa. Testosterone propionate is cheap because we sell a lot of steroids. In addition, we also provide domestic delivery service, which can save your time and make you safer.

Many bodybuilders and fitness enthusiasts buy steroid powders from us, which saves them a lot of money than buying finished products online. If your order is large, we promise that you can purchase testosterone propionate at a price lower than the market price. Long-term win-win cooperation enables us to stand out from many suppliers. I wouldn’t say our site is the best place to buy testosterone propionate, but the top 10 is well deserved.

The advantages of Testosterone Propionate

Testosterone propionate is an anabolic steroid. First, testosterone propionate is good for normal growth and is also useful for the development of male sex organs. Second, it also helps maintain secondary sexual characteristics. Testosterone binds to androgen receptors and, in addition to helping reduce fat, helps muscle growth and repair. Most testosterone products boost immunity, boost energy, increase fat loss, promote good health, and boost libido. If your testosterone levels are low, taking testosterone propionate can bring them back to normal. It helps to gain and maintain lean muscle mass and also prevents osteoporosis.

The half-life of Testosterone Propionate

Testosterone Enanthate has a half-life of about 7 days. Testosterone Cypionate has a half-life of about 6 days. Testosterone Propionate has a half-life of about 2-3 days. Testosterone Propionate needs To inject every day or every other day. The greater volume of injections men when using testosterone propionate is not likable for some users. Now you can understand according to most people choose testosterone Enanthate and Testosterone Cypionate.

Testosterone Propionate dosage

In medicine, testosterone propionate is used to treat androgen deficiency (hypogonadism or androgen withdrawal) in adult males. It is recommended to take 25mg 2-3 times a week.

Testosterone propionate is also used, though rarely, as adjunctive therapy in women with breast cancer. It is not recommended to do so again.

In order to improve physical fitness and performance, the dose of testosterone propionate should be adjusted according to your actual needs. The initial dose of testosterone propionate is usually 300mg per week, especially the first anabolic steroid cycle (this is usually equivalent to 75 to 125mg every other day). Even a minimum of 300 milligrams, with the proper adjustment and rigor of nutrition and training for beginners, can result in some significant improvements in physique and strength. The intermediate dose of testosterone propionate is typically 500-700 mg per week (i.e., 125-175 mg every other day). Some intermediate users are known to be at slightly higher risk, but if the individual’s nutrition and training ingredients are well structured, there are usually not many side effects. Advanced testosterone propionate doses are usually not higher than intermediate cycle doses, but it has been used by athletes up to 700-1000 milligrams per week. Remember, increased testosterone propionate dosage is always associated with increased aromatization and increased severity of side effects.

Testosterone Propionate reviews

Testosterone propionate, which has a short half-life but is cheap, is better suited to bodybuilders who want a quick fix than testosterone. Multiple injections and needles are inevitable and don’t be sad because it’s the sacrifice that makes your muscles grow.

 


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What is Exemestane

Exemestane is a drug used to treat menopausal women breast cancer.

You may have heard of Aromasin, this is the most famous brand. There are many other brands of Exemestane also have the same dose.

Men with breast cancer can take Exemestane, while another called the drug tamoxifen is more commonly used.

How does Exemestane work

Exemestane is to reduce the effect of estrogen in the body. Exemestane belongs to a class of aromatase inhibitors. Exemestane is a kind of aromatase inhibitors. This means it blocks aromatase, an enzyme that converts androgens (hormones produced by the adrenal glands) into estrogen, which is found in the body’s muscles, skin, breasts and fat.

Exemestane Usage

Exemestane is suitable for postmenopausal women estrogen receptor-positive breast cancer patients. If your cancer is hormone-receptor-negative, there is no benefit to Exemestane.

Exemestane Dosage

Exemestane 25mg every day is suggested.

Exemestane is usually taken after the surgery, in order to reduce the risk of breast cancer recurrence or diffusion.

If you are undergoing chemotherapy or radiotherapy, your specialist will tell you the best time to start taking Exemestane.

Sometimes, Exemestane can be used as the first therapy for breast cancer, for example, when the surgery is not appropriate or need to delay. It is sometimes used to shrink larger breast cancers before surgery.

Exemestane can also be used for the treatment of recurrent breast cancer. It can also be used to treat breast cancer (secondary breast cancer) that has spread to other parts of the body, often in combination with another drug.

How long will it take

It depends on your personal circumstances, but Exemestane usually takes 5 to 10 years.

Some people are taking hormone therapy drug Tamoxifen, a few years, Exemestane came into use.

If you’re using it to treat a relapse or if breast cancer has spread to other parts of the body, as long as it controls cancer, you’ll usually take it.

What should I know about drug storage and disposal?

Keep the medicine in a container and keep it sealed away from children. Store at room temperature, away from excess heat and moisture (don’t store in the bathroom).

Exemestane for men

Aromatase inhibitor Exemestane can effectively slow down the boy’s physiological maturity, improve adult male testosterone levels, therefore, aromatase inhibitors can be used to increase the gonads hormone-dependent precocious puberty, idiopathic short and constitutional delayed puberty boy adult height.

Exemestane is better than tamoxifen

A new study finds Aromasin is more effective than Tamoxifen in reducing the risk of breast cancer recurrence, but not all clinicians believe the positive findings. Overall, no cancer survival rates have improved significantly (Exemestane91.1 Tamoxifen87.3 %, %).

 


Off-Season Cycle


If you don’t know steroids, don’t use them lightly. Athletes use steroids to achieve their ideal physique, but it’s not a one-size-fits-all experience. You may get some great muscle for a while, but it’s all in vain if you don’t maintain it during the off-season.

What is a typical off-season cycle like for some of the larger competitive bodybuilders (heavyweight or super-heavyweight)?

Admittedly, everyone’s situation is different, but once a certain level of development is reached, some constants emerge.

Testosterone is the basis of most big men — because we’re talking about the off-season, usually enanthate or cypionate — by about 1,200 to 2,000 milligrams a week. Testosterone is any cycle of bread and butter.

Then there are the anabolic drugs, with most large people taking 600-1000 milligrams of Boldenone or Deca Durabolin (Nandrolone) per week. Sometimes they use Primobolan or Trenbolone, but that’s not common in the offseason; Most people stick to Boldenone and Nandrolone Decanoate, alternating between the two drugs for 8-10 weeks at a time.

After that, you look at the daily dose of growth hormone (4-10 international units per day). Personally, I don’t think it’s necessary to walk higher, although some people will run more if they can afford it.

Most people (but not all) also use insulin, usually 10-20 units per day of humulin-r or Humalog. Again, this is something that some people will use more of, but I don’t think it’s wise from a health standpoint – even from a growth standpoint.

After that, some people might take strange oral steroids from time to time, like Dianabol or Anadrol every few months or so for four weeks, but that’s not really necessary — some people just like a quick boost of strength and bloating.

Most people also take some form of the anti-estrogen drugs, such as Arimidex, throughout the year, about one milligram every other day.


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What is Methenolone Enanthate?

Methenolone Enanthate is an anabolic androgen based on DHT. It is an ester derivative of methenolone and is commonly sold under the brand name Primobolan Depot. When it interacts with aromatase, it doesn’t form any estrogen. It is used by people who are very prone to estrogenic side effects and has lower estrogenic properties than Nandrolone. Metenolone, in the form of enanthate and acetate, can be used as an injection or oral preparation, respectively.

The injection is considered to have high bioavailability. It’s a long-lasting enanthate. It also has a higher survival rate because it bypasses liver failure on its first pass. Methenolone is not 17- -alkylated, but 1- methylated oral bioavailability. This not only reduces stress on the liver but also reduces its availability. A dose of 200 mg or less per week (intramuscular) rarely changes blood pressure.

The application of Primobolan Depot Methenolone Enanthate

Primobolan Depot represents a more popular anabolic steroid in performance-enhancing circles, especially fitness, as Arnold Schwarzenegger’s disgrace surrounds it. Methenolone Enanthate steroid is a mild steroid in the field of bodybuilding.

Primoplan can also be a good steroid for exercise enhancement. It has the ability to promote strength and will have a positive effect on muscular endurance and recovery. Equally important, as it is not a strong mass builder, this can make it a great choice for many athletes. Many athletes simply don’t want to gain too much weight. In some cases, increasing quality can hinder performance. What’s more, staying away from fast-growing muscle mass will protect athletes from prying and suspicious eyes.

Primobolan Depot Dosage

For men, 350-600mg/week, and women, 100mg/week, Primobolan Enanthate’s active life was 10-14 days, and the detection time was about 4-5 weeks. The standard dose for men will drop to 100-200 milligrams a week. The initial treatment typically starts at 200 milligrams per week and is reduced to 100 milligrams per week over time. In some cases, the dose may be reduced by 100 milligrams every two weeks. For male athletes, 300 milligrams per week is generally considered the lowest dose. However, 200 mg/week would provide catabolic protection during the cutting phase, but 300 mg/week would be more effective. Since this is a relatively mild anabolic steroid, most men will find that they can tolerate 400-500 milligrams a week well. For most men, even 600 milligrams a week should be within limits. Weekly doses of more than 600 mg are not uncommon, but keep in mind that doses of less than or more than 600 mg may exacerbate the androgenic activity of steroids. It is generally recommended for 8 to 12 weeks, regardless of the total dose. In terms of stacking, Primobolan can stack well with the vast majority of anabolic steroids. Because it is most commonly used in the cutting phase, steroids such as Anavar, Masteron, Trenbolone, and Winstrol are common additives.

Methenolone Enanthate Reviews

Primobolan, an injectable steroid called methenolone, has long been considered one of the safest steroids. Primobolan depot allows methenolone to be released slowly in the body. Primobolan depot is a moderate anabolic agent with very low androgen levels. The anabolic effect is comparable to that of Deca Durabolin, although the androgen side effects are much less severe. Athletes and bodybuilders will take Primobolan to build muscle. During the Primobolan cycle, your muscle mass will slowly improve. You can expect to keep the gains for several months after the completion of the cycle.


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Buy raw tadalafil powder from us, we are domestic steroid powder supplier in Canada, USA, UK, EU. If you are keen on making steroid from powder, we would provide steroid powder recipe for you.

What is Cialis 

Cialis is the brand name of his Tadalafil, a drug used to treat erectile dysfunction. It is similar to Viagra and Levitra. Under the trade name Adcirca, tadalafil is used for pulmonary hypertension.

Cialis increases the blood flow to the penis, which allows men to erect. It does not cause sexual arousal. It should be used with caution and only under medical supervision.

Tadalafil was approved by the US Food and Drug Administration (FDA) in 2003 for the treatment of erectile dysfunction (ED). It is also used to treat pulmonary hypertension and benign prostatic hyperplasia, enlargement of the prostate gland, leading to urination problems.

How to take Tadalafil?

Tadalafil is usually taken once a day. Follow all instructions on the prescription label. Do not take more or fewer medications or take longer than recommended.

Tadalafil can be taken with or without food.

Don’t destroy or split the Cialis tablet. Swallow it whole.

For erectile dysfunction, take Cialis before sex, but not more than once a day. It can last up to 36 hours before sex. When sexual stimulation occurs, Cialis can help achieve an erection.

If you are taking Adcirca for pulmonary hypertension, do not take Cialis for erectile dysfunction.

Store at room temperature, away from dampness and high temperature.

How fast does Tadalafil work?

Viagra and Levitra take about 30 minutes to work, and the effect lasts about four hours after you take the medicine. You should spend at least two hours before you plan to have sex. After taking it, the effect may last 36 hours.


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Exemestane is a steroid suicide aromatase inhibitor/irreversible aromatase inactivator that reduces estrogen production by blocking aromatase. The medical use of exemestane, like most aromatase inhibitors, is to treat estrogen-dependent breast cancer. It is usually used only when treatment with less aggressive compounds does not produce the desired effect, such as selective estrogen receptor modulators.

For strength athletes and bodybuilders, exemestane has several beneficial characteristics. First, it is reported that exemestane can reduce estrogen by an average of 85%. Of course, doing so helps prevent estrogen-related side effects caused by aromatic steroids. The drug also increases testosterone levels in users, which may be beneficial if used in post-cycle treatment. In addition, there is some evidence that exemestane may increase the level of insulin growth factor (IGF).

Like other aromatase inhibitors, information and Research on the effects of exemestane on lipid/cholesterol in users are conflicting. Some studies have shown that the compound has little effect, while others consider it rather harsh.

Exemestane Dosage

The peak plasma concentration of exemestane was reached within 2 hours after oral administration of 25 mg. The effective life of the drug ranges from 24 to 30 hours. This is important because it is much shorter than non-steroidal inhibitors. A single oral dose of 25 mg of exemestane resulted in a relatively long-term decrease in estrogen levels in plasma and urine. The maximum inhibition occurred about 2 to 3 days after administration and lasted for about 4 to 5 days.

Studies have shown that 25 mg of exemestane is almost as effective as 50 mg in inhibiting estrogen, increasing testosterone and insulin-like growth factor levels. Therefore, the daily dose should not exceed 25 mg. Because of the activity of the compound exemestane, it is administered approximately every 24 hours.

The only negative aspect of the compound seems to be that it takes about seven days to reach a stable plasma level in terms of drug delivery plans. However, this is not the main obstacle to its use. It simply requires users to start using exemestane a week before they expect the compound to be fully effective.

Risk of using exemestane

There was no significant toxicity of exemestane at a daily dose of 600 mg. Most users are well tolerated, and the maximum tolerable dose toxicity has not yet been determined. Negative side effects associated with the use of this compound are usually mild and may include transient gastrointestinal reactions, hot flashes, nausea and/or fatigue. As mentioned earlier, due to conflicting studies, the effect of exemestane on lipid/cholesterol is not yet clear, so monitoring should be carried out when using the compound. Sexual dysfunction is also possible due to lower estrogen levels. However, there are relatively few reports on this aspect.

Because of the minor side effects associated with this compound and its effectiveness in reducing estrogen-related side effects in aromatic steroid synthesis, exemestane seems to be a relatively safe choice in the search for aromatase inhibitors.